Inhibitors?Screening Libraries?ProteinsMedChemExpressTGR5 agonist 1Cat . No.:HY-149807分子式:C??H??NNaO?S分子量:549.74作用靶点:G protein-coupled B ile Acid Receptor 1作用通路:GPCR/G Protein储存方式:Please store the produ ct under the recommended conditions in the Certificate of Analysi s.BIOLOGICAL ACTIVITY生物活性TGR5 agonist 1 (compound 18) 是一种有效的 TGR5 激动剂,EC50 值为 0.31 μM [1]。IC50 & TargetIC50: 0.31 μM (TGR5) [1]REF ERENCESLuxenburger A, et al. The discovery of 12β-methyl-17-epi-1 8-nor-bile acids as potent and selective TGR5 agonists. Eur J Med Chem. 2023 Mar 15;250:115143.McePdfHeightCaution: Product has no t been fully validated for medical applications.For research use only.1/1Master of Bioactive Molecules — 您身边的抑制剂大师 |
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