二、国家自然科学奖 (一) 项目名称 类药性骨架化合物库构建及创新药物发现研究 提名者 中国科学技术协会 完成人 柳红(中国科学院上海药物研究所),周宇(中国科学院上海药物研究所),王江(中国科学院上海药物研究所),郑明月(中国科学院上海药物研究所),陈凯先(中国科学院上海药物研究所) (完成单位) 代表性论文(专著)目录 序号 论文(专著) 名称/刊名/作者 1 Structure-Based Design of Antiviral Drug Candidates Targeting the SARS-CoV-2 Main Protease/Science/ Wenhao Dai#, Bing Zhang#, Xia-Ming Jiang#, Haixia Su#, Jian Li, Yao Zhao, Xiong Xie, Zhenming Jin, Jingjing Peng, Fengjiang Liu, Chunpu Li, You Li, Fang Bai, Haofeng Wang, Xi Cheng, Xiaobo Cen, Shulei Hu, Xiuna Yang, Jiang Wang, Xiang Liu, Gengfu Xiao, Hualiang Jiang, Zihe Rao, Lei-Ke Zhang*, Yechun Xu*, Haitao Yang*, Hong Liu*. 2 Palladium-Catalysed C(sp3)-H Glycosylation for Synthesis of C-Alkyl Glycoamino Acids/Angewandte Chemie International Edition/Yichu Liu, Yibing Wang, Wenhao Dai, Wei Huang, Yingxia Li* and Hong Liu*. 3 Recyclable Ligands for the Non-Enzymatic Dynamic Kinetic Resolution of Challenging α-Amino Acids/Angewandte Chemie International Edition/Yong Nian, Jiang Wang, Shengbin Zhou, Shuni Wang, Hiroki Moriwaki, Aki Kawashima, Vadim A. Soloshonok* and Hong Liu*. 4 Structural optimization and biological evaluation of 1,5-disubstituted pyrazole-3-carboxamines as potent inhibitors of human 5-lipoxygenase/Acta Pharmaceutica Sinica B/Yu Zhou#, Jun Liu#, Mingyue Zheng#, Shuli Zheng, Chunyi Jiang, Xiaomei Zhou, Dong Zhang, Jihui Zhao, Deju Ye, Mingfang Zheng, Hualiang Jiang, Dongxiang Liu*, Jian Cheng* and Hong Liu*. 5 A series of α-heterocyclic carboxaldehyde thiosemicarbazones inhibit topoisomerase IIα catalytic activity/Journal of Medicinal Chemistry/He Huang#, Qin Chen#,Xin Ku, Linghua Meng*, Liping Lin, Xiang Wang, Caihua Zhu, Yi Wang, Zhi Chen, Ming Li, Hualiang Jiang, Kaixian Chen, Jian Ding, Hong Liu*. (二) 项目名称 最优化计算方法和理论 提名者 中国科学技术协会 完成人 戴彧虹(中国科学院数学与系统科学研究院),刘歆(中国科学院数学与系统科学研究院),刘亚锋(中国科学院数学与系统科学研究院) (完成单位) 代表性论文(专著)目录 序号 论文(专著) 名称/刊名/作者 1 A Nonlinear Conjugate Gradient Algorithm with an Optimal Property and an Improved Wolfe Line Search / SIAM Journal on Optimization / YU-HONG DAI and CAI-XIA KOU 2 A Perfect Example for the BFGS Method / Mathematical Programming / Yu-Hong Dai 3 Limited Memory Block Krylov Subspace Optimization for Computing Dominant Singular Value Decompositions / SIAM Journal on Scientific Computing / XIN LIU, ZAIWEN WEN, AND YIN ZHANG 4 All Real Eigenvalues of Symmetric Tensors / SIAM Journal on Matrix Analysis and Applications /CHUN-FENG CUI, YU-HONG DAI, AND JIAWANG NIE 5 Coordinated Beamforming for Miso Interference Channel: Complexity Analysis and Efficient Algorithms / IEEE Transactions on Signal Processing / Ya-Feng Liu, Yu-Hong Dai, and Zhi-Quan Luo (三) 项目名称 T细胞免疫的触发机制 提名者 中国科学技术协会 完成人 许琛琦(中国科学院分子细胞科学卓越创新中心),杨魏(中国科学院分子细胞科学卓越创新中心),施小山(中国科学院分子细胞科学卓越创新中心),吴微(中国科学院分子细胞科学卓越创新中心),李伯良(中国科学院分子细胞科学卓越创新中心) (完成单位) 代表性论文(专著)目录 序号 论文(专著) 名称/刊名/作者 1 Ca2+ regulates T-cell receptor activation by modulating the charge property of lipids/Nature/Xiaoshan Shi,Yunchen Bi,Wei Yang,Xingdong Guo,Yan Jiang,Chanjuan Wan,Lunyi Li,Yibing Bai,Jun Guo,Yujuan Wang,Xiangjun Chen,Bo Wu,Hongbin Sun,Wanli Liu,Junfeng Wang,Chenqi Xu 2 Lipid-dependent conformational dynamics underlie the functional versatility of T-cell receptor/Cell Research/Xingdong Guo,Chengsong Yan,Hua Li,Wenmao Huang,Xiaoshan Shi,Min Huang,Yingfang Wang,Weiling Pan,Mingjun Cai,Lunyi Li,Wei Wu,Yibing Bai,Chi Zhang,Zhijun Liu,Xinyan Wang,Xiaohui F Zhang,Chun Tang,Hongda Wang,Wanli Liu,Bo Ouyang,Catherine C Wong,Yi Cao,Chenqi Xu 3 Potentiating the antitumour response of CD8(+) T cells by modulating cholesterol metabolism/Nature/ Wei Yang,Yibing Bai,Ying Xiong,Jin Zhang,Shuokai Chen,Xiaojun Zheng,Xiangbo Meng,Lunyi Li,Jing Wang,Chenguang Xu,Chengsong Yan,Lijuan Wang,Catharine C. Y. Chang,Ta-Yuan Chang,Ti Zhang,Penghui Zhou,Bao-Liang Song,Wanli Liu,Shao-cong Sun,Xiaolong Liu,Bo-liang Li, Chenqi Xu 4 Multiple signaling roles of CD3e and its application in CAR-T cell therapy/Cell/Wei Wu,Qiuping Zhou,Takeya Masubuchi,Xiaoshan Shi,Hua Li,Xinyi Xu,Min Huang,Li Meng,Xing He,Hengyu Zhu,Shuaixin Gao,Nan Zhang,Ruirui Jing,Jie Sun,Haopeng Wang,Enfu Hui,Catherine Chiulan Wong,Chenqi Xu 5 FBXO38 mediates PD-1 ubiquitination and regulates anti-tumour immunity of T cells/Nature/ Xiangbo Meng,Xiwei Liu,Xingdong Guo,Shutan Jiang,Tingting Chen,Zhiqiang Hu,Haifeng Liu,Yibing Bai,Manman Xue,Ronggui Hu,Shao-cong Sun,Xiaolong Liu,Penghui Zhou,Xiaowu Huang,Lai Wei,Wei Yang,Chenqi Xu (四) 项目名称 发现宇宙早期发光最亮、中心黑洞质量最大的类星体 提名者 中国科学技术协会 完成人 吴学兵(北京大学),王飞格(北京大学),王然(北京大学),易卫敏(中国科学院云南天文台),左文文(中国科学院上海天文台) (完成单位) 代表性论文(专著)目录 序号 论文(专著) 名称/刊名/作者 1 An ultraluminous quasar with a twelve-billion-solar-mass black hole at redshift 6.30 / Nature / Wu, Xue-Bing; Wang, Feige; Fan, Xiaohui; Yi, Weimin; Zuo, Wenwen; Bian, Fuyan; Jiang, Linhua; McGreer, Ian D.; Wang, Ran; Yang, Jinyi; Yang, Qian; Thompson, David; Beletsky, Yuri 2 Probing the Interstellar Medium and Star Formation of the Most Luminous Quasar at z = 6.3/Astrophysical Journal/Wang, Ran; Wu, Xue-Bing; Neri,Roberto; Fan, Xiaohui; Walter, Fabian; Carilli, Chris L.; Momjian, Emmanuel; Bertoldi,Frank; Strauss, Michael A.; Li, Qiong; Wang,Feige; Riechers, Dominik A.; Jiang, Linhua; Omont, Alain;Wagg, Jeff; Cox, Pierre 3 A Survey of Luminous High-redshift Quasars with SDSS and WISE. I. Target Selection and Optical Spectroscopy/Astrophysical Journal/Wang, Feige; Wu, Xue-Bing; Fan, Xiaohui; Yang, Jinyi; Yi, Weimin; Bian, Fuyan; McGreer, Ian D.; Yang, Qian; Ai, Yanli; Dong, Xiaoyi; Zuo, Wenwen; Jiang, Linhua; Green, Richard; Wang, Shu; Cai, Zheng; Wang, Ran; Yue, Minghao 4 SDSS Quasars in the WISE Preliminary Data Release and Quasar Candidate Selection with Optical/Infrared Colors/Astronomical Journal / Wu, Xue-Bing; Hao, Guoqiang; Jia, Zhendong; Zhang, Yanxia; Peng, Nanbo 5 Quasar candidate selection and photometric redshift estimation based on SDSS and UKIDSS data / Monthly Notices of the Royal Astronomical Society / Wu, Xue-Bing; Jia, Zhendong (五) 项目名称 埃迪卡拉纪复杂生物起源和早期演化 提名者 中国科学技术协会 完成人 袁训来(中国科学院南京地质古生物研究所),陈哲(中国科学院南京地质古生物研究所),周传明(中国科学院南京地质古生物研究所),万斌(中国科学院南京地质古生物研究所),华洪(西北大学) (完成单位) 代表性论文(专著)目录 序号 论文(专著) 名称/刊名/作者 1 An early Ediacaran assemblage of macroscopic and morphologically differentiated eukaryotes/ Nature/ Xunlai Yuan, Zhe Chen, Shuhai Xiao, Chuanming Zhou, Hong Hua 2 Death march of a segmented and trilobate bilaterian elucidates early animal evolution/ Nature/ Zhe Chen, Chuanming Zhou, Xunlai Yuan, Shuhai Xiao 3 Cell differentiation and germ-soma separation in Ediacaran animal embryo-like fossils/Nature/ Lei Chen, Shuhai Xiao, Ke Pang, Chuanming Zhou, Xunlai Yuan 4 中国埃迪卡拉纪综合地层和时间框架/中国科学: 地球科学/周传明, 袁训来, 肖书海, 陈哲, 华洪 5 Systematic description of putative animal fossils from the early Ediacaran Lantian Formation of South China/ Palaeontology/Bin Wan, Xunlai Yuan, Zhe Chen, Chengguo Guan, Ke Pang, Qing Tang, Shuhai Xiao (六) 项目名称 面向双高储能器件的新型电极材料的结构设计与性能调控 提名者 中国科学技术协会 完成人 黄富强(中国科学院上海硅酸盐研究所),林天全(中国科学院上海硅酸盐研究所),毕辉(中国科学院上海硅酸盐研究所),董武杰(中国科学院上海硅酸盐研究所) (完成单位) 代表性论文(专著)目录 序号 论文(专著) 名称/刊名/作者 1 Nitrogen-doped mesoporous carbon of extraordinary capacitance for electrochemical energy storage/ Science/ Lin, Tianquan; Chen, I-Wei; Liu, Fengxin; Yang, Chongyin; Bi, Hui; Xu, Fangfang; Huang, Fuqiang. 2 Core-Shell Nanostructured 'Black' Rutile Titania as Excellent Catalyst for Hydrogen Production Enhanced by Sulfur Doping/Journal of the American Chemical Society/Yang, Chongyin; Wang, Zhou; Lin, Tianquan; Yin, Hao; Lü, Xujie; Wan, Dongyun; Xu, Tao; Zheng, Chong; Lin, Jianhua; Huang, Fuqiang; Xie, Xiaoming; Jiang, Mianheng. 3 Visible-light photocatalytic, solar thermal and photoelectrochemical properties of aluminium-reduced black titania/ Energy & Environmental Science / Zhou Wang, Chongyin Yang, Tianquan Lin, Hao Yin, Ping Chen, Dongyun Wan, Fangfang Xu, Fuqiang Huang, Jianhua Lin, Xiaoming Xie, Mianheng Jiang 4 Well-dispersed ruthenium in mesoporous crystal TiO2 as an advanced electrocatalyst for hydrogen evolution reaction/ Journal of the American Chemical Society/ Nong, Shuying; Dong, Wujie; Yin, Junwen; Dong, Bowei; Lu, Yue; Yuan, Xiaotao; Wang, Xin; Bu, Kejun; Chen, Mingyang; Jiang, Shangda; Liu, Li-Min; Sui, Manling; Huang, Fuqiang. 5 A new tubular graphene form of a tetrahedrally connected cellular structure/Advanced Materials/Bi, Hui; Chen, I-Wei; Lin, Tianquan; Huang, Fuqiang. (七) 项目名称 高空核爆炸辐射环境现象学 提名者 中国科学技术协会 完成人 王建国(西北核技术研究所),左应红(西北核技术研究所),牛胜利(西北核技术研究所),朱金辉(西北核技术研究所),陶应龙(西北核技术研究所) (完成单位) 代表性论文(专著)目录 序号 论文(专著) 名称/刊名/作者 1 UNIPIC code for simulations of high power microwave devices/ Physics of Plasmas/ Jianguo Wang, Dianhui Zhang, Chunliang Liu, Yongdong Li, Yue Wang, Hongguang Wang, Hailiang Qiao, and Xiaoze Li 2 高空核爆炸效应参数手册/ 原子能出版社/ 王建国, 牛胜利, 张殿辉, 乔登江 3 Simulation of high-altitude nuclear electromagnetic pulse using a modified model of scattered gamma/ IEEE Transactions on Nuclear Science / Ya Li, Jianguo Wang , Yinghong Zuo, Jinhui Zhu, and Ruyu Fan 4 典型甚低频电磁波对辐射带高能电子的散射损失效应/ 物理学报/ 罗旭东, 牛胜利, 左应红 5 高空核爆炸瞬发辐射电离效应的数值模拟/ 物理学报/ 陶应龙, 王建国, 牛胜利, 朱金辉, 范如玉 |
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